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5HMK

HDM2 in complex with a 3,3-Disubstituted Piperidine

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0043066biological_processnegative regulation of apoptotic process
A0051726biological_processregulation of cell cycle
B0005634cellular_componentnucleus
B0043066biological_processnegative regulation of apoptotic process
B0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 62Q A 1001
ChainResidue
ALEU54
AHIS96
AILE99
ATYR100
BLYS51
B62Q1001
ALEU57
AGLY58
AILE61
AMET62
ATYR67
AGLN72
APHE91
AVAL93

site_idAC2
Number of Residues17
Detailsbinding site for residue 62Q B 1001
ChainResidue
ALYS51
AGLU52
ATYR55
A62Q1001
BGLN24
BLEU54
BLEU57
BGLY58
BILE61
BMET62
BTYR67
BGLN72
BPHE91
BVAL93
BHIS96
BILE99
BTYR100

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues166
DetailsDomain: {"description":"SWIB/MDM2","evidences":[{"source":"PROSITE-ProRule","id":"PRU01273","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

242842

PDB entries from 2025-10-08

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