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5HM0

Crystal structure of the first bromodomain of human BRD4 bound to benzoisoxazoloazepine 3

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 62V A 201
ChainResidue
APRO53
AHOH353
ATRP81
APRO82
ALEU92
ALYS99
AASN140
AASP145
AILE146
AHOH317

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

222036

PDB entries from 2024-07-03

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