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5HJP

Identification of LXRbeta selective agonists for the treatment of Alzheimer's Disease

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0003707molecular_functionnuclear steroid receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0008270molecular_functionzinc ion binding
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006629biological_processlipid metabolic process
C0003677molecular_functionDNA binding
C0003707molecular_functionnuclear steroid receptor activity
C0005634cellular_componentnucleus
C0006355biological_processregulation of DNA-templated transcription
C0008270molecular_functionzinc ion binding
D0003677molecular_functionDNA binding
D0004879molecular_functionnuclear receptor activity
D0006629biological_processlipid metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues19
Detailsbinding site for residue 668 B 501
ChainResidue
BASN239
BARG319
BPHE329
BLEU330
BLEU345
BPHE349
BHIS435
BGLN438
BLEU442
BLEU449
BTRP457
BSER242
BTHR272
BLEU274
BALA275
BILE277
BGLU281
BMET312
BTHR316

site_idAC2
Number of Residues3
Detailsbinding site for residue PEG B 502
ChainResidue
BVAL218
BGLN219
BLEU220

site_idAC3
Number of Residues2
Detailsbinding site for residue PEG C 601
ChainResidue
BPRO251
CLYS478

site_idAC4
Number of Residues18
Detailsbinding site for residue 668 D 501
ChainResidue
DASN239
DPHE268
DTHR272
DLEU274
DALA275
DILE277
DSER278
DMET312
DTHR316
DARG319
DPHE329
DLEU330
DLEU345
DPHE349
DHIS435
DGLN438
DLEU442
DTRP457

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0000269|PubMed:20159957
ChainResidueDetails
BLYS410
BLYS448
DLYS410
DLYS448

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PDB entries from 2024-07-24

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