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5GTR

estrogen receptor alpha in complex with a stabilized peptide antagonist 6

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue EST A 601
ChainResidue
ALEU346
ALEU525
AALA350
AGLU353
ALEU387
AMET388
ALEU391
AARG394
AMET421
AHIS524

site_idAC2
Number of Residues9
Detailsbinding site for residues IAS C 2 and DPP C 5
ChainResidue
ALYS416
AGLU542
CARG1
CILE3
C0JY4
CARG6
C0JY7
CGLN9
CNH210

site_idAC3
Number of Residues12
Detailsbinding site for residues 0JY C 4 and DPP C 5
ChainResidue
AILE358
AVAL376
AGLU542
AMET543
CARG1
CIAS2
CILE3
CARG6
C0JY7
C0JY8
CGLN9
CNH210

site_idAC4
Number of Residues11
Detailsbinding site for residues 0JY C 7 and 0JY C 8
ChainResidue
AVAL355
AILE358
ALYS362
ALEU372
AGLN375
ALEU379
CILE3
C0JY4
CDPP5
CARG6
CGLN9

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ATYR537

site_idSWS_FT_FI2
Number of Residues1
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447

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PDB entries from 2024-07-24

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