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5GTP

The agonist-free structure of human PPARgamma ligand binding domain in the presence of the SRC-1 coactivator peptide

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue MYR A 501
ChainResidue
APHE226
AMET329
APHE363
AGOL502
AHOH625
ACYS285
AARG288
ASER289
AALA292
AGLU295
AILE296
AILE326
ATYR327

site_idAC2
Number of Residues8
Detailsbinding site for residue GOL A 502
ChainResidue
APHE282
AGLN286
ASER289
AHIS323
APHE363
AHIS449
ATYR473
AMYR501

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
BSER698
AHIS323
AHIS449
ATYR473

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224

237423

PDB entries from 2025-06-11

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