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5GTN

Human PPARgamma ligand binding dmain complexed with R35

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues21
Detailsbinding site for residue Q35 A 501
ChainResidue
ALYS263
ASER289
AHIS323
ALEU330
AMET334
AILE341
AMET364
APHE368
AHIS449
ALEU469
ATYR473
APHE264
AHOH693
AHOH761
AARG280
AILE281
APHE282
AGLY284
ACYS285
AGLN286
AARG288

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
BSER698
AHIS323
AHIS449
ATYR473

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224

222415

PDB entries from 2024-07-10

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