5G3J
Discovery of New Selective Glucocorticoid Receptor Agonist Leads
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE CPS A 1777 |
Chain | Residue |
A | TRP610 |
A | ASP638 |
A | ASP641 |
A | TYR660 |
A | TYR735 |
A | MET745 |
site_id | AC2 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO A 1778 |
Chain | Residue |
A | HOH2020 |
A | HOH2021 |
A | PRO541 |
A | TRP577 |
A | LYS667 |
site_id | AC3 |
Number of Residues | 15 |
Details | BINDING SITE FOR RESIDUE E7T A 1779 |
Chain | Residue |
A | MET560 |
A | LEU563 |
A | ASN564 |
A | GLN570 |
A | TRP600 |
A | MET601 |
A | MET604 |
A | ARG611 |
A | PHE623 |
A | GLN642 |
A | MET646 |
A | THR739 |
A | PHE749 |
A | LEU753 |
A | HOH2033 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | CROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530 |
Chain | Residue | Details |
A | LYS703 |