Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

5FP8

Crystal structure of human KDM4D in complex with 3-4-methylthiophen-2- ylmethylaminopyridine-4-carboxylic acid

Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 350
ChainResidue
ACYS238
AHIS244
ACYS310
ACYS312

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CO A 360
ChainResidue
AHOH2354
AHIS192
AGLU194
AHIS280
AAUY1341
AHOH2347

site_idAC3
Number of Residues11
DetailsBINDING SITE FOR RESIDUE AUY A 1341
ChainResidue
AHIS90
ATYR136
AASP139
APHE189
AHIS192
ALYS210
ATRP212
AHIS280
ACO360
AHOH2347
AHOH2354

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1342
ChainResidue
APRO113
ALYS124
AASN128
ATRP185
ALYS186
AHOH2288

site_idAC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 1343
ChainResidue
AARG60
AGLU61
ATHR62
AHOH2158
AHOH2161
AHOH2488
AHOH2489

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1344
ChainResidue
AARG123
ALYS124
ALYS127
AASN128

site_idAC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1345
ChainResidue
AARG102
AHIS103
AASN106
AHOH2231
AHOH2238

site_idAC8
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1346
ChainResidue
AGLN116
AGLN116
AASN117
AASN117

site_idAC9
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 1347
ChainResidue
AASP302
ATYR303
AMET306

site_idBC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1348
ChainResidue
ATYR181
AGLU194
AALA292
AHOH2297
AHOH2347

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues42
DetailsDomain: {"description":"JmjN","evidences":[{"source":"PROSITE-ProRule","id":"PRU00537","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues166
DetailsDomain: {"description":"JmjC","evidences":[{"source":"PROSITE-ProRule","id":"PRU00538","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"B2RXH2","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues3
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU00538","evidenceCode":"ECO:0000255"},{"source":"PubMed","id":"26741168","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"PDB","id":"5F5A","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5F5C","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues2
DetailsModified residue: {"description":"PolyADP-ribosyl glutamic acid","evidences":[{"source":"PubMed","id":"23102699","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

PDB statisticsPDBj update infoContact PDBjnumon