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5FG5

Crystal structure of the bromodomain of human BRPF1 in complex with PFI-4 chemical probe

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 5XF A 801
ChainResidue
AILE635
AHOH917
AILE652
AGLU655
AVAL657
APRO658
AGLU661
AASN708
APHE714
AHOH906

site_idAC2
Number of Residues2
Detailsbinding site for residue NO3 B 801
ChainResidue
BPRO632
BPHE633

site_idAC3
Number of Residues12
Detailsbinding site for residue 5XF B 802
ChainResidue
BILE635
BLYS639
BASN651
BILE652
BPHE653
BGLU655
BVAL657
BPRO658
BGLU661
BASN708
BPHE714
BHOH907

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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