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5FDO

Mcl-1 complexed with small molecule inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
C0042981biological_processregulation of apoptotic process
D0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 5X2 A 400
ChainResidue
APHE228
ALEU267
APHE270
AGLY271
AILE294
BASN223
BHIS224
AMET231
ALEU246
AMET250
AVAL253
AASN260
AGLY262
AARG263
ATHR266

site_idAC2
Number of Residues13
Detailsbinding site for residue 5X2 B 400
ChainResidue
AASN223
AHIS224
BPHE228
BMET231
BLEU246
BMET250
BASN260
BGLY262
BARG263
BTHR266
BLEU267
BPHE270
BGLY271

site_idAC3
Number of Residues10
Detailsbinding site for residue 5X2 C 400
ChainResidue
CHIS224
CPHE228
CMET231
CMET250
CVAL253
CARG263
CTHR266
CLEU267
CPHE270
CGLY271

site_idAC4
Number of Residues13
Detailsbinding site for residue 5X2 D 400
ChainResidue
DALA227
DPHE228
DMET231
DLEU246
DVAL249
DMET250
DVAL253
DGLY262
DARG263
DTHR266
DLEU267
DPHE270
DGLY271

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
ALYS194
DLYS194
DLYS197
ALYS197
BLYS194
BLYS197
CLYS194
CLYS197

222036

PDB entries from 2024-07-03

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