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5FC4

Mcl-1 complexed with small molecule inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue 5WL A 401
ChainResidue
AALA227
ALEU267
APHE270
A5WL402
A5WL402
A5WK403
AHOH521
AHOH640
APHE228
AMET231
AVAL249
AMET250
AGLY262
AARG263
AARG263
ATHR266

site_idAC2
Number of Residues13
Detailsbinding site for residue 5WL A 402
ChainResidue
ATHR191
AALA227
ALYS234
ALEU235
AVAL249
AHIS252
AVAL253
AASP256
A5WL401
A5WL401
AHOH570
AHOH605
AHOH609

site_idAC3
Number of Residues12
Detailsbinding site for residue 5WK A 403
ChainResidue
AARG176
AALA202
AGLY203
AARG207
AARG215
AGLY262
AVAL265
ATHR266
APHE319
A5WL401
AHOH522
AHOH608

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvaqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
ALYS194
ALYS197

221371

PDB entries from 2024-06-19

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