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5FBK

Crystal structure of the extracellular domain of human calcium sensing receptor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004930molecular_functionG protein-coupled receptor activity
A0007186biological_processG protein-coupled receptor signaling pathway
A0016020cellular_componentmembrane
B0004930molecular_functionG protein-coupled receptor activity
B0007186biological_processG protein-coupled receptor signaling pathway
B0016020cellular_componentmembrane
Functional Information from PROSITE/UniProt
site_idPS00979
Number of Residues19
DetailsG_PROTEIN_RECEP_F3_1 G-protein coupled receptors family 3 signature 1. VaNLLgLFyIPQVSyASSS
ChainResidueDetails
AVAL153-SER171

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues166
DetailsRegion: {"description":"Ligand-binding 1 (LB1)","evidences":[{"source":"PubMed","id":"17360426","evidenceCode":"ECO:0000303"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues16
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"34194040","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27386547","evidenceCode":"ECO:0000305"},{"source":"PDB","id":"5FBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5FBK","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3E","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3F","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3G","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"34194040","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"38326620","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27386547","evidenceCode":"ECO:0000305"},{"source":"PDB","id":"5FBK","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3E","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3F","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3G","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8SZF","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"34194040","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"38326620","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27386547","evidenceCode":"ECO:0000305"},{"source":"PDB","id":"5FBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5FBK","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3E","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3F","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7M3G","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8SZF","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"34467854","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5K5T","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7E6T","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27386547","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"33603117","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"34194040","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"5FBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5FBK","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7DTU","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27386547","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"33603117","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"34194040","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"38326620","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"5FBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5FBK","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7DTU","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7DTV","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8SZG","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27386547","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"33603117","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"34194040","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"38326620","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"5FBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5FBK","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7DTU","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8SZG","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI10
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"34467854","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"7E6T","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI11
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"33603117","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"34467854","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7DTT","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"7E6T","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI12
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"38326620","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8SZF","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI13
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27386547","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"5FBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5FBK","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"5K5S","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI14
Number of Residues2
DetailsSite: {"description":"Important for ability of agonist AMG 416 to activate G-protein-coupled receptor activity","evidences":[{"source":"PubMed","id":"26290606","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI15
Number of Residues5
DetailsGlycosylation: {"description":"N-linked (GlcNAc...) asparagine","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI16
Number of Residues10
DetailsGlycosylation: {"description":"N-linked (GlcNAc...) asparagine","evidences":[{"evidenceCode":"ECO:0000255"},{"source":"PubMed","id":"27434672","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"33603117","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"7DTT","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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