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5F1H

Crystal structure of the BRD9 bromodamian in complex with BI-9564.

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 5U6 A 201
ChainResidue
AHIS42
ATYR106
AHOH303
AHOH350
AGLY43
APHE44
APHE45
APHE47
AVAL49
AILE53
AALA54
AASN100

site_idAC2
Number of Residues11
Detailsbinding site for residue 5U6 B 201
ChainResidue
BHIS42
BPHE44
BPHE45
BPHE47
BPRO48
BVAL49
BILE53
BASN100
BTYR106
BHOH301
BHOH341

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsRegion: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsSite: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

242500

PDB entries from 2025-10-01

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