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5F0C

Structure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium tuberculosis in complex with compound 4 at 1.87A resolution

Functional Information from GO Data
ChainGOidnamespacecontents
A0000976molecular_functiontranscription cis-regulatory region binding
A0003677molecular_functionDNA binding
A0003700molecular_functionDNA-binding transcription factor activity
A0005515molecular_functionprotein binding
A0005829cellular_componentcytosol
A0006355biological_processregulation of DNA-templated transcription
A0045892biological_processnegative regulation of DNA-templated transcription
A0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 5TE A 301
ChainResidue
ATHR121
ATRP207
ATRP138
AMET142
ATRP145
ATHR149
AASN176
AASN179
AGLU180
ALEU183

site_idAC2
Number of Residues3
Detailsbinding site for residue SO4 A 302
ChainResidue
AASP98
AARG99
AHOH421

site_idAC3
Number of Residues6
Detailsbinding site for residue SO4 A 303
ChainResidue
APRO41
ALEU42
AALA123
AALA126
AHOH404
AHOH408

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues19
DetailsDNA_BIND: H-T-H motif => ECO:0000255|PROSITE-ProRule:PRU00335
ChainResidueDetails
ASER46-PHE65

site_idSWS_FT_FI2
Number of Residues2
DetailsSITE: Inhibitor-binding
ChainResidueDetails
AASN176
AASN179

223532

PDB entries from 2024-08-07

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