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5EP3

Quorum-Sensing Signal Integrator LuxO - Catalytic Domain Bound to CV-133 Inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0005524molecular_functionATP binding
A0006355biological_processregulation of DNA-templated transcription
A0008134molecular_functiontranscription factor binding
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 5QT A 401
ChainResidue
AGLY141
AGLN363
APHE142
AILE143
ATHR174
AGLY175
AVAL178
AARG316
AILE323
AVAL359

site_idAC2
Number of Residues7
Detailsbinding site for residue SO4 A 402
ChainResidue
AGLU171
AGLY173
ATHR174
AGLY175
ALYS176
AHOH505
AHOH579

site_idAC3
Number of Residues15
Detailsbinding site for residue EPE A 403
ChainResidue
ALYS163
AALA164
ATHR165
AILE258
AGLN259
AVAL274
AASP275
AVAL276
AVAL305
AGLU351
AARG367
AHOH510
AHOH529
AHOH553
AHOH627

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 404
ChainResidue
ASER158
ALYS337
AVAL371
ATHR374
AHOH614

Functional Information from PROSITE/UniProt
site_idPS00676
Number of Residues16
DetailsSIGMA54_INTERACT_2 Sigma-54 interaction domain ATP-binding region B signature. GaVemAHNGTLMLDEL
ChainResidueDetails
AGLY228-LEU243

site_idPS00688
Number of Residues10
DetailsSIGMA54_INTERACT_3 Sigma-54 interaction domain C-terminal part signature. WPGNVRELqN
ChainResidueDetails
ATRP355-ASN364

222624

PDB entries from 2024-07-17

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