5EK9
Crystal structure of the second bromodomain of human BRD2 in complex with a tetrahydroquinoline inhibitor
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 9 |
Details | binding site for residue 5P4 A 501 |
Chain | Residue |
A | TRP370 |
A | PRO371 |
A | PHE372 |
A | LEU381 |
A | LEU383 |
A | CYS425 |
A | ASN429 |
A | HIS433 |
A | HOH617 |
site_id | AC2 |
Number of Residues | 7 |
Details | binding site for residue 5P4 B 501 |
Chain | Residue |
B | TRP370 |
B | PRO371 |
B | LEU381 |
B | ASN429 |
B | ASP434 |
B | HOH602 |
B | HOH647 |
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 60 |
Details | BROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY |
Chain | Residue | Details |
A | ALA369-TYR428 |