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5EK0

Human Nav1.7-VSD4-NavAb in complex with GX-936.

Functional Information from GO Data
ChainGOidnamespacecontents
A0005216molecular_functionmonoatomic ion channel activity
A0005261molecular_functionmonoatomic cation channel activity
A0005886cellular_componentplasma membrane
A0006811biological_processmonoatomic ion transport
A0016020cellular_componentmembrane
A0055085biological_processtransmembrane transport
B0005216molecular_functionmonoatomic ion channel activity
B0005261molecular_functionmonoatomic cation channel activity
B0005886cellular_componentplasma membrane
B0006811biological_processmonoatomic ion transport
B0016020cellular_componentmembrane
B0055085biological_processtransmembrane transport
C0005216molecular_functionmonoatomic ion channel activity
C0005261molecular_functionmonoatomic cation channel activity
C0005886cellular_componentplasma membrane
C0006811biological_processmonoatomic ion transport
C0016020cellular_componentmembrane
C0055085biological_processtransmembrane transport
D0005216molecular_functionmonoatomic ion channel activity
D0005261molecular_functionmonoatomic cation channel activity
D0005886cellular_componentplasma membrane
D0006811biological_processmonoatomic ion transport
D0016020cellular_componentmembrane
D0055085biological_processtransmembrane transport
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue PX4 A 1801
ChainResidue
ALEU1654
APHE1655
ATYR1694
APRO1695
ATYR1696
DARG1599

site_idAC2
Number of Residues7
Detailsbinding site for residue PX4 A 1802
ChainResidue
APHE1670
ATYR1671
BPRO1695
BTRP1698
ATHR1665
AGLY1667
AGLU1668

site_idAC3
Number of Residues1
Detailsbinding site for residue PX4 A 1804
ChainResidue
AGLN1618

site_idAC4
Number of Residues3
Detailsbinding site for residue PX4 A 1807
ChainResidue
AGLN1530
AGLU1534
A5P21808

site_idAC5
Number of Residues16
Detailsbinding site for residue 5P2 A 1808
ChainResidue
AGLU1534
ATYR1537
ATRP1538
AASN1540
AVAL1541
AGLY1581
AMET1582
APHE1583
AALA1585
AASP1586
APHE1598
AARG1602
AALA1604
AARG1605
AARG1608
APX41807

site_idAC6
Number of Residues6
Detailsbinding site for residue PX4 B 1801
ChainResidue
ATHR1596
AARG1599
BTYR1694
BPRO1695
BTYR1696
BALA1697

site_idAC7
Number of Residues8
Detailsbinding site for residue PX4 B 1802
ChainResidue
BTHR1665
BGLY1667
BGLU1668
BPHE1670
BTYR1671
CMET1691
CPRO1695
CTRP1698

site_idAC8
Number of Residues1
Detailsbinding site for residue PX4 B 1803
ChainResidue
BGLN1618

site_idAC9
Number of Residues1
Detailsbinding site for residue PX4 B 1804
ChainResidue
BMET1677

site_idAD1
Number of Residues3
Detailsbinding site for residue PX4 B 1805
ChainResidue
BGLU1534
BASP1586
B5P21806

site_idAD2
Number of Residues15
Detailsbinding site for residue 5P2 B 1806
ChainResidue
BGLU1534
BTYR1537
BTRP1538
BASN1540
BVAL1541
BGLY1581
BMET1582
BPHE1583
BALA1585
BASP1586
BPHE1598
BARG1602
BARG1605
BARG1608
BPX41805

site_idAD3
Number of Residues4
Detailsbinding site for residue PX4 C 1801
ChainResidue
BTHR1596
CTYR1694
CPRO1695
CTYR1696

site_idAD4
Number of Residues7
Detailsbinding site for residue PX4 C 1802
ChainResidue
CTYR1645
CTHR1665
CGLY1667
CGLU1668
CPHE1670
DTYR1696
DTRP1698

site_idAD5
Number of Residues1
Detailsbinding site for residue PX4 C 1803
ChainResidue
CGLN1618

site_idAD6
Number of Residues3
Detailsbinding site for residue PX4 C 1804
ChainResidue
CGLU1534
CTRP1538
C5P21805

site_idAD7
Number of Residues16
Detailsbinding site for residue 5P2 C 1805
ChainResidue
CTYR1537
CTRP1538
CASN1540
CGLY1581
CMET1582
CPHE1583
CALA1585
CASP1586
CGLU1589
CTHR1590
CPHE1598
CARG1602
CALA1604
CARG1605
CARG1608
CPX41804

site_idAD8
Number of Residues6
Detailsbinding site for residue PX4 D 1801
ChainResidue
ATRP1698
DPHE1644
DGLY1667
DGLU1668
DPHE1670
AMET1691

site_idAD9
Number of Residues5
Detailsbinding site for residue PX4 D 1802
ChainResidue
CARG1599
DPHE1655
DTYR1694
DPRO1695
DTYR1696

site_idAE1
Number of Residues2
Detailsbinding site for residue PX4 D 1805
ChainResidue
DGLU1534
D5P21806

site_idAE2
Number of Residues17
Detailsbinding site for residue 5P2 D 1806
ChainResidue
DGLU1534
DTYR1537
DTRP1538
DASN1540
DVAL1541
DSER1578
DGLY1581
DMET1582
DPHE1583
DALA1585
DASP1586
DPHE1598
DARG1602
DALA1604
DARG1605
DARG1608
DPX41805

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues72
DetailsTOPO_DOM: Extracellular => ECO:0000305|PubMed:30765606
ChainResidueDetails
AGLU1524-GLU1534
AILE1588-THR1596
BGLU1524-GLU1534
BILE1588-THR1596
CGLU1524-GLU1534
CILE1588-THR1596
DGLU1524-GLU1534
DILE1588-THR1596

237423

PDB entries from 2025-06-11

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