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5DY7

Crystal structure of the human BRPF1 bromodomain in complex with SEED4

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue 5GT A 801
ChainResidue
AILE652
AVAL657
APRO658
AGLU661
AVAL662
AASN708
APHE714
AHOH917
AHOH929

site_idAC2
Number of Residues8
Detailsbinding site for residue NO3 A 802
ChainResidue
ASER702
ALEU705
ALYS706
ATYR715
AVAL719
AARG722
AHOH915
AHOH987

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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