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5DW1

X-ray crystal structure of human BRD2(BD2) in complex with RVX297 to 1.55 A resolution

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 5GD A 500
ChainResidue
ATRP370
DHOH636
APRO371
APHE372
AVAL376
ALEU381
ALEU383
AASN429
AHIS433
AHOH626

site_idAC2
Number of Residues13
Detailsbinding site for residue 5GD B 500
ChainResidue
BPRO371
BPHE372
BVAL376
BLEU381
BLEU383
BASN429
BHIS433
BVAL435
BHOH616
BHOH630
CHOH629
CHOH643
CHOH689

site_idAC3
Number of Residues14
Detailsbinding site for residue 5GD C 501
ChainResidue
BTRP370
BALA380
CTRP370
CPRO371
CPHE372
CVAL376
CLEU381
CASN429
CHIS433
CHOH625
CHOH651
CHOH672
CHOH690
DHIS384

site_idAC4
Number of Residues5
Detailsbinding site for residue NA C 502
ChainResidue
CASP377
CSER379
CHOH679
CHOH712
CHOH719

site_idAC5
Number of Residues14
Detailsbinding site for residue 5GD D 501
ChainResidue
ATRP370
AALA380
BSER379
BHIS384
DPRO371
DPHE372
DVAL376
DLEU381
DLEU383
DASN429
DHIS433
DHOH630
DHOH678
DHOH701

site_idAC6
Number of Residues6
Detailsbinding site for residue NA D 502
ChainResidue
AHOH661
AHOH671
AHOH699
BHOH646
DGLY382
DHOH683

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

222415

PDB entries from 2024-07-10

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