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5DVC

Human PPARgamma ligand binding dmain complexed with SB1453 in a covalent bonded form

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues19
Detailsbinding site for residue T53 A 501
ChainResidue
AILE262
AILE326
AILE341
ASER342
AGLU343
APHE363
ALEU453
ALEU469
ATYR473
AHOH607
AHOH665
APHE264
AILE267
APHE282
AGLY284
ACYS285
AGLN286
AARG288
ASER289

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
BSER698
AHIS323
AHIS449
ATYR473

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224

237735

PDB entries from 2025-06-18

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