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5D7X

Crystal structure of the human BRPF1 bromodomain in complex with XZ08

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue NO3 A 801
ChainResidue
AGLY650
AILE652
ALEU688
AASN689
AALA717
AARG720
AHOH917
AHOH1027

site_idAC2
Number of Residues12
Detailsbinding site for residue XZ8 A 802
ChainResidue
APHE653
AGLU655
APRO656
AVAL657
APRO658
AASN708
APHE714
AHOH928
AHOH939
AHOH959
AHOH1038
AILE652

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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