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5CQ3

Crystal structure of the bromodomain of bromodomain adjacent to zinc finger domain protein 2B (BAZ2B) in complex with 6-Hydroxypicolinic acid (SGC - Diamond I04-1 fragment screening)

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue EDO A 2001
ChainResidue
AMET1875
AGLU1879
ALYS1964
ATHR1968

site_idAC2
Number of Residues7
Detailsbinding site for residue EDO A 2002
ChainResidue
ADMS2004
APO42005
ALYS1896
ALEU1897
AVAL1898
APRO1899
A53B2003

site_idAC3
Number of Residues7
Detailsbinding site for residue 53B A 2003
ChainResidue
AASN1944
AILE1950
AEDO2002
APO42005
AHOH2102
AHOH2104
AHOH2132

site_idAC4
Number of Residues5
Detailsbinding site for residue DMS A 2004
ChainResidue
ASER1948
AASP1949
AILE1950
AEDO2002
AHOH2175

site_idAC5
Number of Residues9
Detailsbinding site for residue PO4 A 2005
ChainResidue
AASN1944
AGLU1945
ASER1948
AEDO2002
A53B2003
AHOH2101
AHOH2102
AHOH2113
AHOH2116

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA1886-PHE1943

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphothreonine => ECO:0007744|PubMed:21406692
ChainResidueDetails
ALEU1918

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:21406692
ChainResidueDetails
ATYR1923

222036

PDB entries from 2024-07-03

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