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5BT5

Crystal structure of BRD2 second bromodomain in complex with SGC-CBP30 chemical probe

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue EDO A 501
ChainResidue
ATYR426
AARG440
AGLN443
AGLN443
AASP444
AGLU447
APHE448
AHOH631

site_idAC2
Number of Residues6
Detailsbinding site for residue EDO A 502
ChainResidue
ALYS402
AASP407
AMET438
ALYS441
AHOH608
ATYR368

site_idAC3
Number of Residues7
Detailsbinding site for residue EDO A 503
ChainResidue
AILE389
AILE390
ALYS391
AHIS392
AASN424
ALYS427
AASP455

site_idAC4
Number of Residues4
Detailsbinding site for residue EDO A 504
ChainResidue
AHIS352
AHIS384
ALYS452
APRO454

site_idAC5
Number of Residues9
Detailsbinding site for residue 2LO A 505
ChainResidue
ATRP370
APRO371
APHE372
AASP377
ALEU383
AASN429
AHIS433
AVAL435
AHOH603

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

222624

PDB entries from 2024-07-17

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