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5AWK

Crystal structure of VDR-LBD/partial agonist complex: 22S-ethyl analogue

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue YSE A 501
ChainResidue
ATYR143
ALEU305
AHIS393
ALEU229
ASER233
AARG270
ASER271
ASER274
ATRP282
AVAL296
AHIS301

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBINDING: BINDING => ECO:0000269|PubMed:15065852, ECO:0000269|PubMed:17227670
ChainResidueDetails
AHIS301
AHIS393
ATYR143
ALEU223
AILE267

219869

PDB entries from 2024-05-15

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