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5AWJ

Crystal structure of VDR-LBD/partial agonist complex: 22S-hexyl analogue

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue YSL A 501
ChainResidue
ATYR143
AVAL296
AHIS301
ALEU305
ALEU389
AHIS393
APHE418
ALEU223
AVAL230
ASER233
AARG270
ASER271
ASER274
ATRP282
ACYS284

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:15065852, ECO:0007744|PDB:1RK3
ChainResidueDetails
ATYR143
ASER233
AARG270
ASER274
AHIS301
AHIS393

224201

PDB entries from 2024-08-28

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