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5ACU

VIM-2-NAT, Discovery of novel inhibitor scaffolds against the metallo- beta-lactamase VIM-2 by SPR based fragment screening

Functional Information from GO Data
ChainGOidnamespacecontents
A0008800molecular_functionbeta-lactamase activity
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE OH A 1001
ChainResidue
AHIS116
AHIS118
AASP120
AHIS196
AZN1296
AZN1297

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE ZN A 1296
ChainResidue
AOH1001
AZN1297
AHIS116
AHIS118
AHIS196

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE ZN A 1297
ChainResidue
AASP120
ACYS221
AHIS263
AOH1001
AZN1296

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1298
ChainResidue
AHIS170
AHIS285
ACL1299
ACL1300

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL A 1299
ChainResidue
AHIS170
AHIS285
AZN1298
AHOH2016

site_idAC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CL A 1300
ChainResidue
AALA135
AHIS170
AZN1298

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PDB entries from 2026-01-14

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