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4Z6H

Crystal structure of BRD9 bromodomain in complex with a valerolactam quinolone ligand

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue 4L2 A 201
ChainResidue
AGLY43
APHE44
APHE45
APHE47
AVAL49
AASN100
ATYR106
AHOH307
BGLU124

site_idAC2
Number of Residues8
Detailsbinding site for residue 4L2 B 201
ChainResidue
BGLY43
BPHE44
BPHE45
BVAL49
BILE53
BASN100
BTYR106
BHOH303

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsRegion: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsSite: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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