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4XY8

Crystal Structure of the bromodomain of BRD9 in complex with a 2-amine-9H-purine ligand

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 43U A 201
ChainResidue
APHE44
AHOH388
APHE47
AVAL49
AILE53
ATYR99
AASN100
ATYR106
AHIS115
AHOH331

site_idAC2
Number of Residues2
Detailsbinding site for residue BR A 202
ChainResidue
AVAL105
ALYS123

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsRegion: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsSite: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

250359

PDB entries from 2026-03-11

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