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4XUA

Crystal Structure of the bromodomain of human BAZ2B in complex with E11919 BAZ2-ICR analogue

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 2001
ChainResidue
AVAL1893
AASN1894
ALEU1895
AHOH2241
AHOH2242
AHOH2280

site_idAC2
Number of Residues3
Detailsbinding site for residue EDO A 2002
ChainResidue
AHIS1883
AGLU1884
AHOH2200

site_idAC3
Number of Residues5
Detailsbinding site for residue EDO A 2003
ChainResidue
AASP1938
AGLU1941
ATHR1942
AHOH2172
AHOH2225

site_idAC4
Number of Residues6
Detailsbinding site for residue EDO A 2004
ChainResidue
AARG1864
ALEU1872
ATHR1968
AHOH2183
AHOH2210
AHOH2303

site_idAC5
Number of Residues16
Detailsbinding site for residue 43C A 2005
ChainResidue
ATRP1887
APRO1888
ALEU1890
ALEU1891
APRO1892
AVAL1893
AASN1894
AVAL1898
ATYR1901
AASN1944
AILE1950
AHOH2129
AHOH2227
AHOH2238
AHOH2277
AHOH2307

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA1886-PHE1943

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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