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4XT9

RORgamma (263-509) complexed with GSK2435341A and SRC2

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues31
DetailsPocket 1 in Model 1 Assembly 1 (Ligand L_LIG_1 ) (Entity 3)
ChainResidue
ACYS285
AALA327
AMET358
AVAL361
AARG364
AMET365
AARG367
AALA368
ATYR369
AVAL376
APHE377
AGLN286
APHE378
AGLU379
APHE388
ALEU391
ACYS393
ALEU396
AILE397
AILE400
APHE401
ASER404
ALEU287
AHIS479
ATYR502
ALEU292
ATRP317
ACYS320
AALA321
AHIS323
ALEU324

site_idAC2
Number of Residues20
DetailsPocket 2 in Model 1 Assembly 1 (Ligand M_SO4_2 ) (Entity 4)
ChainResidue
AGLU359
ATYR420
ALEU423
AVAL424
AILE426
AASN427
AHIS429
AARG430
APRO431
AGLN443
AGLU447
APHE450
AHIS451
ALEU463
ALEU466
APRO467
APRO468
ALYS469
ALEU472
AARG473

site_idAC3
Number of Residues17
DetailsPocket 3 in Model 1 Assembly 1
ChainResidue
ALEU289
ALEU293
AARG296
ACYS366
AARG367
AALA368
ATYR369
AASN370
AALA371
AASP372
ALEU407
ASER408
ALEU410
AHIS411
APHE412
AGLU414
AILE417

site_idAC4
Number of Residues15
DetailsNeighbourhood of 1:B_LYS_688 _B_ILE_689 _B_LEU_690 _B_HIS_691 _B_ARG_692 _B_LEU_693 _B_LEU_694 _B_GLN_695 (Entity 2)
ChainResidue
AGLU504
ALEU501
APRO500
AHOH716
ALEU353
AILE350
ALEU505
ALYS354
AVAL332
AGLN346
ALYS336
AHOH735
AGLN349
AMET342
APHE341

site_idAC5
Number of Residues26
DetailsNeighbourhood of 1:L_LIG_1 (Entity 3)
ChainResidue
AVAL376
ALEU324
ACYS320
AHIS479
AMET358
AILE400
APHE388
APHE401
ASER404
AILE397
AGLN286
AHOH727
AMET365
AVAL361
AARG364
ACYS285
AHOH725
AARG367
ALEU292
ALEU287
AALA368
AHOH724
APHE377
AHOH733
APHE378
AHIS323

site_idAC6
Number of Residues15
Detailsbinding site for residue 43V A 601
ChainResidue
ACYS285
AGLN286
ALEU287
ALEU292
ACYS320
AHIS323
AARG364
AARG367
AALA368
APHE377
APHE378
APHE388
AILE400
APHE401
AHOH724

site_idAC7
Number of Residues4
Detailsbinding site for residue SO4 A 602
ChainResidue
AARG310
ALYS469
AGLY470
ASO4603

site_idAC8
Number of Residues4
Detailsbinding site for residue SO4 A 603
ChainResidue
ALYS311
APRO468
ALYS469
ASO4602

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PDB entries from 2024-07-24

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