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4XF7

myo-inositol 3-kinase bound with its substrates (AMPPCP and myo-inositol)

Functional Information from GO Data
ChainGOidnamespacecontents
A0000166molecular_functionnucleotide binding
A0016301molecular_functionkinase activity
B0000166molecular_functionnucleotide binding
B0016301molecular_functionkinase activity
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue INS A 301
ChainResidue
AASP12
AASP219
AHOH448
AHOH456
AGLY25
AGLY26
AGLY27
ATYR30
ATYR75
AGLN136
AARG140
ATHR215

site_idAC2
Number of Residues26
Detailsbinding site for residue ACP A 302
ChainResidue
AASN83
AARG85
AHIS164
AASP166
ASER187
AASN188
AGLY189
APRO190
APHE204
APRO206
AVAL207
AVAL209
ASER214
AGLY216
AALA217
AGLY218
ATHR245
ALEU249
AMG303
AHOH426
AHOH428
AHOH430
AHOH435
AHOH447
AHOH448
AHOH456

site_idAC3
Number of Residues6
Detailsbinding site for residue MG A 303
ChainResidue
AGLN136
AACP302
AHOH426
AHOH435
AHOH447
AHOH448

site_idAC4
Number of Residues3
Detailsbinding site for residue IOD A 304
ChainResidue
AGLU59
ALEU64
AHOH411

site_idAC5
Number of Residues2
Detailsbinding site for residue IOD A 305
ChainResidue
ATHR203
AGLU269

site_idAC6
Number of Residues4
Detailsbinding site for residue IOD A 308
ChainResidue
AASP101
AIOD309
BGLN236
BIOD310

site_idAC7
Number of Residues2
Detailsbinding site for residue IOD A 309
ChainResidue
AIOD308
BIOD310

site_idAC8
Number of Residues1
Detailsbinding site for residue IOD A 310
ChainResidue
BGLU146

site_idAC9
Number of Residues1
Detailsbinding site for residue IOD A 311
ChainResidue
ALEU99

site_idAD1
Number of Residues4
Detailsbinding site for residue IOD A 312
ChainResidue
ALEU99
ASER123
AALA124
ALYS127

site_idAD2
Number of Residues2
Detailsbinding site for residue IOD A 313
ChainResidue
AARG85
AILE147

site_idAD3
Number of Residues1
Detailsbinding site for residue IOD A 315
ChainResidue
AVAL235

site_idAD4
Number of Residues10
Detailsbinding site for residue INS B 301
ChainResidue
BASP12
BGLY25
BGLY26
BGLY27
BTYR30
BTYR75
BGLN136
BARG140
BASP219
BHOH428

site_idAD5
Number of Residues21
Detailsbinding site for residue ACP B 302
ChainResidue
BARG85
BHIS164
BASP166
BSER187
BASN188
BGLY189
BPHE204
BVAL207
BVAL209
BSER214
BALA217
BGLY218
BTHR245
BLEU249
BMG303
BHOH417
BHOH419
BHOH424
BHOH426
BHOH428
BHOH432

site_idAD6
Number of Residues6
Detailsbinding site for residue MG B 303
ChainResidue
BHOH426
BHOH428
BGLN136
BACP302
BHOH423
BHOH424

site_idAD7
Number of Residues1
Detailsbinding site for residue IOD B 304
ChainResidue
BTHR203

site_idAD8
Number of Residues2
Detailsbinding site for residue IOD B 305
ChainResidue
BARG11
BPRO51

site_idAD9
Number of Residues1
Detailsbinding site for residue IOD B 306
ChainResidue
BSER123

site_idAE1
Number of Residues1
Detailsbinding site for residue IOD B 307
ChainResidue
BPRO144

site_idAE2
Number of Residues1
Detailsbinding site for residue IOD B 308
ChainResidue
BHOH415

site_idAE3
Number of Residues4
Detailsbinding site for residue IOD B 310
ChainResidue
AASP101
AIOD308
AIOD309
BLYS239

site_idAE4
Number of Residues4
Detailsbinding site for residue IOD B 311
ChainResidue
AGLU98
ALEU99
APRO100
BGLN236

site_idAE5
Number of Residues2
Detailsbinding site for residue IOD B 312
ChainResidue
BASP182
BTYR229

site_idAE6
Number of Residues2
Detailsbinding site for residues IOD B 309 and IOD B 313
ChainResidue
AARG85
BTYR170

220113

PDB entries from 2024-05-22

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