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4WMR

STRUCTURE OF MCL1 BOUND TO BRD inhibitor ligand 1 AT 1.7A

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue ZN A 401
ChainResidue
AHIS224
A865404
APOP405

site_idAC2
Number of Residues3
Detailsbinding site for residue ZN A 402
ChainResidue
AHIS252
AASP256
APOP406

site_idAC3
Number of Residues2
Detailsbinding site for residue ZN A 403
ChainResidue
APOP405
APOP405

site_idAC4
Number of Residues18
Detailsbinding site for residue 865 A 404
ChainResidue
ATHR226
AALA227
ALEU246
AMET250
AVAL253
AARG263
ATHR266
ALEU267
APHE270
AGLY271
AZN401
APOP405
APOP405
AHOH560
AHOH584
AHOH587
AHOH601
AHIS224

site_idAC5
Number of Residues10
Detailsbinding site for residue POP A 405
ChainResidue
AHIS224
AZN401
AZN403
AZN403
A865404
A865404
AHOH512
AHOH518
AHOH560
AHOH601

site_idAC6
Number of Residues7
Detailsbinding site for residue POP A 406
ChainResidue
ASER172
AHIS252
AASP256
AARG300
AZN402
AHOH540
AHOH617

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues14
DetailsMotif: {"description":"BH3"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues20
DetailsMotif: {"description":"BH1"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues15
DetailsMotif: {"description":"BH2"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues3
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)"}
ChainResidueDetails

251174

PDB entries from 2026-03-25

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