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4WLB

Crystal structure of RORc in complex with a partial inverse agonist compound

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue 3QQ A 601
ChainResidue
ACYS285
AALA368
APHE378
APHE388
ALEU396
AILE397
AILE400
AHIS479
AHOH885
AGLN286
ALEU287
ATRP317
ACYS320
AHIS323
AARG364
AMET365
AARG367

site_idAC2
Number of Residues14
Detailsbinding site for residue TLA A 602
ChainResidue
AARG294
AASN298
AHOH721
AHOH725
AHOH741
AHOH882
AHOH892
AHOH912
BSER301
BGLU303
BGLU304
BTHR457
BHIS458
BARG459

site_idAC3
Number of Residues10
Detailsbinding site for residue TLA A 603
ChainResidue
AARG296
AALA371
ASER408
AHIS411
AHOH716
AHOH737
AHOH771
BARG374
BHIS405
BHOH703

site_idAC4
Number of Residues17
Detailsbinding site for residue 3QQ B 601
ChainResidue
BCYS285
BGLN286
BLEU287
BTRP317
BCYS320
BHIS323
BARG364
BARG367
BALA368
BPHE378
BPHE388
BLEU396
BILE400
BPHE401
BHIS479
BHOH768
BHOH794

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PDB entries from 2025-06-11

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