Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4UX4

Crystal structure of human tankyrase 2 in complex with 1-methyl-7-(4- methylphenyl)-5-oxo-5,6-dihydro-1,6-naphthyridin-1-ium

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE E9L B 2162
ChainResidue
BHIS1031
BGLU1138
BGLY1032
BPHE1035
BTYR1050
BTYR1060
BALA1062
BLYS1067
BSER1068
BTYR1071

site_idAC2
Number of Residues9
DetailsBINDING SITE FOR RESIDUE E9L A 2162
ChainResidue
AHIS1031
AGLY1032
ATYR1050
ATYR1060
AALA1062
ALYS1067
ASER1068
ATYR1071
AGLU1138

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 2163
ChainResidue
BCYS1081
BHIS1084
BCYS1089
BCYS1092

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 2163
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC5
Number of Residues9
DetailsBINDING SITE FOR RESIDUE SO4 A 2164
ChainResidue
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070
AHOH4043
AHOH4047
AHOH4146
AHOH4207

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 2164
ChainResidue
BARG977
BHIS979
BARG980
BLYS1067
BGLN1070
BHOH4033
BHOH4146

site_idAC7
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 2165
ChainResidue
BASN990
BARG991
BPRO1160
BGLU1161
BHOH4045
BHOH4165

site_idAC8
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 2165
ChainResidue
AASN990
AARG991
APRO1160
AGLU1161
AHOH4062
AHOH4065

site_idAC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 2166
ChainResidue
AARG1128
APRO1129
ASER1130
AVAL1131
AASN1132
AGLY1133

site_idBC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE GOL B 2166
ChainResidue
BARG977
BHIS979
BGLY983
BGLY987
BILE988
BPHE989
BHOH4042
BHOH4043

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092
BCYS1081
BHIS1084
BCYS1089
BCYS1092

222624

PDB entries from 2024-07-17

PDB statisticsPDBj update infoContact PDBjnumon