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4UDD

GR in complex with desisobutyrylciclesonide

Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE CPS A 1778
ChainResidue
ATRP610
AGLN776
ALYS777
AHOH2236
AHOH2237
AHOH2238
AHOH2239
AASP641
AGLN642
ATYR660
AASN731
ATYR735
AGLN738
AMET745
AILE747

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CPS A 1779
ChainResidue
ATYR640
AHIS645
ATYR648
AGLU727
AHOH2088
AHOH2242

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CPS A 1780
ChainResidue
AMET691
ALYS695
AVAL702
ASER708
ATRP712
APHE715

site_idAC4
Number of Residues8
DetailsBINDING SITE FOR RESIDUE EDO A 1781
ChainResidue
AGLU540
APRO541
ATRP577
AMET604
ALYS667
AHOH2011
AHOH2042
AHOH2043

site_idAC5
Number of Residues14
DetailsBINDING SITE FOR RESIDUE CV7 A 1782
ChainResidue
AMET560
ALEU563
AASN564
AGLY567
AGLN570
AARG611
AMET646
ATYR735
ACYS736
ATHR739
AILE747
APHE749
AHOH2044
AHOH2084

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues165
DetailsRegion: {"description":"Interaction with CRY1","evidences":[{"source":"PubMed","id":"22170608","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO)","evidences":[{"source":"PubMed","id":"12144530","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 3"}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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