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4TYL

Fragment-Based Screening of the Bromodomain of ATAD2

Functional Information from GO Data
ChainGOidnamespacecontents
A0006325biological_processchromatin organization
A0006355biological_processregulation of transcription, DNA-templated
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue SO4 A 1201
ChainResidue
AARG987
AARG990
AARG994
AARG1067
AARG1072
AHOH1302

site_idAC2
Number of Residues3
Detailsbinding site for residue CL A 1202
ChainResidue
AARG1077
AHOH1352
AHOH1365

site_idAC3
Number of Residues7
Detailsbinding site for residue 39O A 1203
ChainResidue
AVAL1008
AVAL1013
ATYR1063
AASN1064
AILE1074
AHOH1407
AHOH1459

site_idAC4
Number of Residues1
Detailsbinding site for residue CL A 1204
ChainResidue
AHOH1366

site_idAC5
Number of Residues4
Detailsbinding site for residue CL A 1205
ChainResidue
AHOH1387
AHOH1387
AHOH1395
AHOH1395

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PDB entries from 2024-03-27

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