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4QNS

Crystal structure of bromodomain from Plasmodium faciparum GCN5, PF3D7_0823300

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
B0004402molecular_functionhistone acetyltransferase activity
C0004402molecular_functionhistone acetyltransferase activity
D0004402molecular_functionhistone acetyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE SO4 A 1501
ChainResidue
ATRP1454
DILE1441
ATYR1457
AGLU1458
AEDO1503
AHOH1606
AHOH1640
AHOH1663
DTHR1439
DTHR1440

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 1502
ChainResidue
AARG1408
AARG1411
AHIS1412

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1503
ChainResidue
AGLY1422
AILE1423
ALYS1426
ATRP1454
ASO41501
DILE1441

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1504
ChainResidue
AGLY1355
AHIS1356
ALYS1357
AGLU1358
AEDO1505

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 1505
ChainResidue
AGLY1355
AHIS1356
AEDO1504
DHOH1702

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 1501
ChainResidue
BGLY1355
BHIS1356
BSO41506
BHOH1735
BHOH1736
BHOH1742

site_idAC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 B 1502
ChainResidue
BARG1408
BARG1411
DLYS1398

site_idAC8
Number of Residues10
DetailsBINDING SITE FOR RESIDUE SO4 B 1503
ChainResidue
BTRP1454
BTYR1457
BGLU1458
BEDO1504
BHOH1636
BHOH1679
BHOH1717
CTHR1439
CTHR1440
CILE1441

site_idAC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 1504
ChainResidue
BGLY1422
BILE1423
BTYR1457
BSO41503
CILE1441

site_idBC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ACT B 1505
ChainResidue
BPRO1380
BASN1436
BTYR1442
BHOH1627

site_idBC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 1506
ChainResidue
BGLY1355
BHIS1356
BLYS1357
BGLU1358
BSO41501
BHOH1719

site_idBC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 C 1501
ChainResidue
CARG1408
CARG1411

site_idBC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 C 1502
ChainResidue
CLYS1426
CTYR1457
CGLU1458
CHOH1633
CHOH1681

site_idBC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO C 1503
ChainResidue
CTYR1394
CASP1395
CLYS1398

site_idBC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO D 1501
ChainResidue
DSER1386
DLEU1387
DSER1388

site_idBC7
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO D 1502
ChainResidue
BHIS1412
BASP1414
DPRO1384
DVAL1385
DTYR1394
DHOH1639

site_idBC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE ACT D 1503
ChainResidue
DGLU1419
DLYS1426
DTYR1457
DGLU1458
DHOH1657

site_idBC9
Number of Residues3
DetailsBINDING SITE FOR RESIDUE ACT D 1504
ChainResidue
DLEU1366
DARG1407
DARG1411

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PDB entries from 2025-07-02

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