4NQN
Crystal Structure of the bromodomain of human BRD9 in complex with a triazolo-phthalazine ligand
Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 10 |
| Details | BINDING SITE FOR RESIDUE Y1Z A 201 |
| Chain | Residue |
| A | HIS42 |
| A | HOH306 |
| A | PHE44 |
| A | PHE45 |
| A | ILE53 |
| A | ASN100 |
| A | TYR106 |
| A | ARG125 |
| A | ALA128 |
| A | SER132 |
Functional Information from SwissProt/UniProt
| site_id | SWS_FT_FI2 |
| Number of Residues | 2 |
| Details | Region: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]} |
| Chain | Residue | Details |
| site_id | SWS_FT_FI3 |
| Number of Residues | 2 |
| Details | Site: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]} |
| Chain | Residue | Details |






