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4NQN

Crystal Structure of the bromodomain of human BRD9 in complex with a triazolo-phthalazine ligand

Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE Y1Z A 201
ChainResidue
AHIS42
AHOH306
APHE44
APHE45
AILE53
AASN100
ATYR106
AARG125
AALA128
ASER132

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI2
Number of Residues2
DetailsRegion: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsSite: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

242199

PDB entries from 2025-09-24

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