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4N10

Crystal structure of plasmodium falciparum oxidized glutaredoxin 1 (PfGrx1) complexed with cisplatin

Functional Information from GO Data
ChainGOidnamespacecontents
A0015038molecular_functionglutathione disulfide oxidoreductase activity
A0016209molecular_functionantioxidant activity
A0016491molecular_functionoxidoreductase activity
A0019153molecular_functionprotein-disulfide reductase (glutathione) activity
A0046872molecular_functionmetal ion binding
A0098869biological_processcellular oxidant detoxification
Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE MPO A 201
ChainResidue
ASER5
AASP89
AHOH301
AHOH316
AHOH331
ALYS9
ATYR31
AASN61
ATYR65
AGLU68
APRO76
AGLY87
ACYS88

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE MPD A 202
ChainResidue
AASN13
AGLU17
ALYS82

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CPT A 203
ChainResidue
AMET59
AGLN63
ALYS93
AHOH321
AHOH354

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CPT A 204
ChainResidue
AMET48
AHIS49
ALYS67
AHOH336
AHOH353

site_idAC5
Number of Residues9
DetailsBINDING SITE FOR RESIDUE CPT A 205
ChainResidue
AASN19
AMET48
AHIS49
AVAL50
ALYS67
AGLU68
AGLY71
AHOH336
AHOH347

Functional Information from PROSITE/UniProt
site_idPS00195
Number of Residues17
DetailsGLUTAREDOXIN_1 Glutaredoxin active site. VFakteCPYCikAisiL
ChainResidueDetails
AVAL23-LEU39

221051

PDB entries from 2024-06-12

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