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4MR5

Crystal Structure of the second bromodomain of human BRD2 in complex with a quinazolinone ligand (RVX-OH)

Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 501
ChainResidue
ATYR368
ALYS402
AASP407
AMET438
ALYS441
AHOH626

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 502
ChainResidue
AGLN443
AASP444
AHOH657
ATYR426
AARG440
AGLN443

site_idAC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 503
ChainResidue
AASP385
ATYR428

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 504
ChainResidue
AILE389
AILE390
ALYS391
AHIS392
AASN424
ALYS427
AASP455

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE DMS A 505
ChainResidue
ATRP370
AHIS433
AHOH691
AHOH694
AHOH695

site_idAC6
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 1K0 A 506
ChainResidue
ALYS351
ATRP370
APRO371
APHE372
AVAL376
ALEU381
ALEU383
AASN429
AHIS433
AHOH604
AHOH691

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

248636

PDB entries from 2026-02-04

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