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4MN3

Chromodomain antagonists that target the polycomb-group methyllysine reader protein Chromobox homolog 7 (CBX7)

Functional Information from GO Data
ChainGOidnamespacecontents
A0035102cellular_componentPRC1 complex
Functional Information from PDB Data
site_idAC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 101
ChainResidue
ALYS25
ATRP29
APRO30

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 102
ChainResidue
ALYS32
AMET49
AGLU52
AHOH203
AHOH232

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 103
ChainResidue
ATRP29
APRO45
BHOH103
ALYS27

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE MG A 104
ChainResidue
AGLU2
AGLU2
AHIS41
AHIS41

site_idAC5
Number of Residues8
DetailsBINDING SITE FOR RESIDUE P33 A 105
ChainResidue
ALYS12
ALYS13
AVAL15
ALEU23
APRO31
ASER34
AGLU55
AHOH222

Functional Information from PROSITE/UniProt
site_idPS00598
Number of Residues21
DetailsCHROMO_1 Chromo domain signature. YlVKWkGWppkys.TWEPeehI
ChainResidueDetails
ATYR22-ILE42

223166

PDB entries from 2024-07-31

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