4MDD
Crystal Structure of the Glucocorticoid Receptor Bound to a Non-steroidal Antagonist Reveals Repositioning and Partial Disordering of Activation Function Helix 12
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 9 |
Details | BINDING SITE FOR RESIDUE 29M A 801 |
Chain | Residue |
A | MET560 |
A | LEU563 |
A | ASN564 |
A | GLN570 |
A | MET604 |
A | ALA605 |
A | LEU608 |
A | CYS736 |
A | THR739 |
site_id | AC2 |
Number of Residues | 11 |
Details | BINDING SITE FOR RESIDUE 29M B 801 |
Chain | Residue |
B | MET560 |
B | LEU563 |
B | ASN564 |
B | GLY567 |
B | GLN570 |
B | MET604 |
B | ALA605 |
B | LEU608 |
B | PHE623 |
B | TYR735 |
B | CYS736 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 4 |
Details | CROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530 |
Chain | Residue | Details |
A | LYS703 | |
B | LYS703 |