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4LVT

Bcl_2-Navitoclax (ABT-263) Complex

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues19
DetailsBINDING SITE FOR RESIDUE 1XJ A 301
ChainResidue
AALA97
AGLY142
AARG143
AVAL145
AALA146
APHE195
ALEU198
ATYR199
AHOH431
AHOH434
AHOH491
AASP100
APHE101
AARG104
ATYR105
AASP108
APHE109
AASN140
ATRP141

site_idAC2
Number of Residues16
DetailsBINDING SITE FOR RESIDUE 1XJ B 301
ChainResidue
BALA97
BASP100
BPHE101
BTYR105
BPHE109
BVAL130
BASN140
BTRP141
BGLY142
BVAL145
BALA146
BVAL153
BPHE195
BLEU198
BTYR199
BHOH456

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues19
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. LFrDGv.NWGRIVAFFeFGG
ChainResidueDetails
ALEU134-GLY152

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WIqdnGGWDaFV
ChainResidueDetails
ATRP185-VAL196

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. VhltLRqAGDDFSRR
ChainResidueDetails
AVAL90-ARG104

site_idPS01260
Number of Residues21
DetailsBH4_1 Apoptosis regulator, Bcl-2 family BH4 motif signature. DNREIVmKYIHYKLSQRGYeW
ChainResidueDetails
AASP8-TRP28

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues40
DetailsMotif: {"description":"BH4","evidences":[{"source":"PROSITE-ProRule","id":"PRU00025","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues28
DetailsMotif: {"description":"BH3","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues38
DetailsMotif: {"description":"BH1","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues30
DetailsMotif: {"description":"BH2","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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