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4KLZ

Inhibition of Small GTPases by Stabilization of the GDP Complex, a Novel Approach applied to Rit1, a Target for Rheumatoid Arthritis

Functional Information from GO Data
ChainGOidnamespacecontents
A0003924molecular_functionGTPase activity
A0005525molecular_functionGTP binding
A0007165biological_processsignal transduction
A0016020cellular_componentmembrane
Functional Information from PDB Data
site_idAC1
Number of Residues17
DetailsBINDING SITE FOR RESIDUE GDP A 501
ChainResidue
AGLY31
ALYS135
AASP137
ALEU138
ASER164
AALA165
AALA166
AMG502
AHOH618
AVAL32
AGLY33
ALYS34
ASER35
AALA36
APHE46
AGLU48
AASN134

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE MG A 502
ChainResidue
ASER35
AGDP501
AHOH618

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AGLY28
AASP75
AASN134

222926

PDB entries from 2024-07-24

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