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4JXH

Complexe of ARNO Sec7 domain with the protein-protein interaction inhibitor N-(4-hydroxy-2,6-dimethylphenyl)benzenesulfonamide at pH 8.5

Functional Information from GO Data
ChainGOidnamespacecontents
A0005085molecular_functionguanyl-nucleotide exchange factor activity
A0032012biological_processregulation of ARF protein signal transduction
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE HRC A 301
ChainResidue
ASER56
AHOH674
ALEU148
AARG152
ALEU153
APRO154
AILE160
AILE245
AHOH574
AHOH647

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PO4 A 302
ChainResidue
AGLY116
AGLN158
ALYS159
AARG162
AHOH664
AHOH684

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues129
DetailsDomain: {"description":"SEC7","evidences":[{"source":"PROSITE-ProRule","id":"PRU00189","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

249697

PDB entries from 2026-02-25

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