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4JNA

Crystal structure of the DepH complex with dimethyl-FK228

Functional Information from GO Data
ChainGOidnamespacecontents
A0000166molecular_functionnucleotide binding
A0016491molecular_functionoxidoreductase activity
B0000166molecular_functionnucleotide binding
B0016491molecular_functionoxidoreductase activity
Functional Information from PDB Data
site_idAC1
Number of Residues39
DetailsBINDING SITE FOR RESIDUE FAD A 401
ChainResidue
AGLY55
AARG82
AARG83
AASN84
ASER90
AHIS91
AASP123
ASER124
AVAL125
AALA153
APHE154
ASER57
AGLY155
AASP158
ACYS180
AHIS181
ASER273
ASER274
AGLY310
AASP311
AGLY317
ATHR318
AHIS58
AVAL319
AHOH505
AHOH506
AHOH517
AHOH520
AHOH531
AHOH545
AHOH551
AHOH578
AHOH647
AALA59
AILE77
AASP78
AALA79
AGLY80
AALA81

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CL A 402
ChainResidue
AHIS176
ACYS177
AHIS181

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 403
ChainResidue
APHE86
AASP158
ALEU160
AGLU167
AHOH539

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 404
ChainResidue
AALA114
ATYR115
BHOH515
BHOH580

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE PO4 A 405
ChainResidue
AVAL238
AARG239
AASP240
AARG257
AHOH532

site_idAC6
Number of Residues38
DetailsBINDING SITE FOR RESIDUE FAD B 401
ChainResidue
BILE54
BGLY55
BSER57
BHIS58
BALA59
BILE77
BASP78
BALA79
BGLY80
BALA81
BARG83
BASN84
BSER90
BHIS91
BASP123
BSER124
BVAL125
BPHE154
BGLY155
BASP158
BCYS180
BHIS181
BSER273
BSER274
BGLY310
BASP311
BGLY317
BTHR318
BVAL319
BCL402
BHOH501
BHOH502
BHOH510
BHOH512
BHOH516
BHOH531
BHOH543
BHOH568

site_idAC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL B 402
ChainResidue
BHIS176
BCYS177
BHIS181
BFAD401

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 403
ChainResidue
AGLN96
BILE94
BGLY95
BGLN96
AILE94

site_idAC9
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO B 404
ChainResidue
AHOH634
BTYR115
BHOH540

site_idBC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL B 405
ChainResidue
BPRO197
BTYR200
BGLN226
BARG241
BALA254

site_idBC2
Number of Residues15
DetailsBINDING SITE FOR CHAIN H OF DIMETHYL FK228
ChainResidue
ALEU328
AILE331
AARG335
BCYS177
BASP255
BARG257
BPRO288
BTHR313
BHIS314
BARG315
BGLY316
HHOH101
HHOH102
HHOH103
HHOH104

site_idBC3
Number of Residues10
DetailsBINDING SITE FOR CHAIN I OF DIMETHYL FK228
ChainResidue
ACYS177
ATYR179
AMET267
AHIS314
AARG315
AGLY316
BLEU328
BILE331
BARG335
IHOH101

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PDB entries from 2024-07-10

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