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4J1P

X-ray crystal structure of bromodomain 2 of human brd2 in complex with rvx208 to 1.08 A resolution

Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE 1K0 A 501
ChainResidue
APRO371
AHOH786
AHOH793
AHOH850
APHE372
AVAL376
ALEU381
AASN429
AHIS433
AHOH604
AHOH644
AHOH754

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 502
ChainResidue
AHOH614
AHOH628
AHOH670
AHOH726
AHOH771

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues109
DetailsDomain: {"description":"Bromo 2","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

243531

PDB entries from 2025-10-22

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