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4IR4

Crystal Structure of the bromodomain of human BAZ2B in complex with 1-[7-(morpholin-4-yl)-1-(pyridin-2-yl)indolizin-3-yl]ethanone (GSK2834113A)

Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE IR4 A 2001
ChainResidue
ATRP1887
APRO1888
APRO1899
AASN1944
AILE1950
AHOH2188

site_idAC2
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 2002
ChainResidue
AHIS1883
AGLU1884

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2003
ChainResidue
ATHR1968
APHE1969
AARG1864

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2004
ChainResidue
AGLU1927
ATRP1965
AHOH2217

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2005
ChainResidue
AVAL1893
AASN1894
ALEU1895
AHOH2110
AHOH2169

site_idAC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2006
ChainResidue
ALYS1903
AGLU1945
AASP1946

site_idAC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2007
ChainResidue
ALYS1907
ALEU1935
AHOH2202

site_idAC8
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 2008
ChainResidue
ALEU1872
AMET1875
AGLU1879
ATHR1968

site_idAC9
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 2009
ChainResidue
ALYS1902
AGLU1945
AASP1947
AHOH2195

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA1886-PHE1943

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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