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4IR3

Crystal Structure of the bromodomain of human BAZ2B in complex with 1-[7-amino-1-(pyrimidin-2-yl)indolizin-3-yl]ethanone (GSK2833282A)

Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE EDO A 2001
ChainResidue
ALYS1917
AGLN1922
APRO1924
ATHR1928
AASP1932
AHOH2177
AHOH2207
AHOH2208

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 2002
ChainResidue
AGLU1945
AASP1947
AHOH2178
AHOH2221
AHOH2222
ALYS1902

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2003
ChainResidue
ALYS1903
AGLU1945
AASP1946

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 2004
ChainResidue
ALYS1906
ALYS1907
APRO1908
AHOH2159
AHOH2194
AHOH2233

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL A 2005
ChainResidue
ATHR1882
AHIS1883
AGLU1884
AHOH2220

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE 1FK A 2006
ChainResidue
ATRP1887
APRO1888
AASN1944
AILE1950
AHOH2176
AHOH2224
AHOH2229

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA1886-PHE1943

221716

PDB entries from 2024-06-26

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