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4IA3

Diastereotopic and Deuterium Effects in Gemini

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE BIV A 501
ChainResidue
ATYR175
ALEU337
ALEU338
AHIS423
ALEU258
ASER265
AARG302
ASER303
ASER306
ATRP314
ACYS316
AHIS333

site_idAC2
Number of Residues15
DetailsBINDING SITE FOR CHAIN B OF NUCLEAR RECEPTOR COACTIVATOR 2
ChainResidue
AILE270
ALYS274
AARG280
AILE288
ALYS292
APRO434
AGLU435
AGLU446
AGLU451
AHOH603
BHOH701
BHOH702
BHOH703
BHOH704
BHOH705

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues18
DetailsRegion: {"description":"Interaction with coactivator LXXLL motif","evidences":[{"source":"UniProtKB","id":"P13053","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"UniProtKB","id":"P11473","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"17218092","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2HC4","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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